Selective PPAR modulator
A selective PPAR modulator (SPPARM) is a selective receptor modulator of the peroxisome proliferator-activated receptor (PPAR).[1][2][3] Examples include SPPARMs of the PPARγ, BADGE, EPI-001, INT-131, MK-0533, and S26948.
See also
- PPAR agonist
References
- ^ Fruchart, Jean-Charles; Santos, Raul D.; Aguilar-Salinas, Carlos; Aikawa, Masanori; Al Rasadi, Khalid; Amarenco, Pierre; Barter, Philip J.; Ceska, Richard; Corsini, Alberto; Després, Jean-Pierre; Duriez, Patrick; Eckel, Robert H.; Ezhov, Marat V.; Farnier, Michel; Ginsberg, Henry N.; Hermans, Michel P.; Ishibashi, Shun; Karpe, Fredrik; Kodama, Tatsuhiko; Koenig, Wolfgang; Krempf, Michel; Lim, Soo; Lorenzatti, Alberto J.; McPherson, Ruth; Nuñez-Cortes, Jesus Millan; Nordestgaard, Børge G.; Ogawa, Hisao; Packard, Chris J.; Plutzky, Jorge; Ponte-Negretti, Carlos I.; Pradhan, Aruna; Ray, Kausik K.; Reiner, Željko; Ridker, Paul M.; Ruscica, Massimiliano; Sadikot, Shaukat; Shimano, Hitoshi; Sritara, Piyamitr; Stock, Jane K.; Su, Ta-Chen; Susekov, Andrey V.; Tartar, André; Taskinen, Marja-Riitta; Tenenbaum, Alexander; Tokgözoğlu, Lale S.; Tomlinson, Brian; Tybjærg-Hansen, Anne; Valensi, Paul; Vrablík, Michal; Wahli, Walter; Watts, Gerald F.; Yamashita, Shizuya; Yokote, Koutaro; Zambon, Alberto; Libby, Peter (4 June 2019). "The selective peroxisome proliferator-activated receptor alpha modulator (SPPARMα) paradigm: conceptual framework and therapeutic potential". Cardiovascular Diabetology. 18 (1): 71. doi:10.1186/s12933-019-0864-7. ISSN 1475-2840. PMC 6549355. PMID 31164165.
- ^ Fruchart, Jean-Charles; Hermans, Michel P.; Fruchart-Najib, Jamila; Kodama, Tatsuhiko (3 January 2021). "Selective Peroxisome Proliferator-Activated Receptor Alpha Modulators (SPPARMα) in the Metabolic Syndrome: Is Pemafibrate Light at the End of the Tunnel?". Current Atherosclerosis Reports. 23 (1): 3. doi:10.1007/s11883-020-00897-x. ISSN 1534-6242. PMC 7779417. PMID 33392801.
- ^ Balint, B. L.; Nagy, L. (March 2006). "Selective modulators of PPAR activity as new therapeutic tools in metabolic diseases". Endocrine, Metabolic & Immune Disorders Drug Targets. 6 (1): 33–43. doi:10.2174/187153006776056620. ISSN 1871-5303. PMID 16611163.
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PPARTooltip Peroxisome proliferator-activated receptor modulators
- Agonists: 15-HETE
- 15-HpETE
- Aleglitazar
- Aluminium clofibrate
- Arachidonic acid
- Bezafibrate
- Chiglitazar
- Clofibrate
- CP-775146
- Daidzein
- DHEA (prasterone) (in rodents)
- Elafibranor
- Etomoxir
- Fenofibrate
- Genistein
- Gemfibrozil
- GW-7647
- Lanifibranor
- Leukotriene B4
- LG-101506
- LG-100754
- Lobeglitazone
- Muraglitazar
- Oleylethanolamide
- Palmitoylethanolamide
- Pemafibrate
- Perfluorononanoic acid
- Perfluorooctanoic acid
- Pioglitazone
- Saroglitazar
- Sodelglitazar
- Tesaglitazar
- Tetradecylthioacetic acid
- Troglitazone
- WY-14643
- Antagonists: GW-6471
- MK-886
- Agonists: 15-HETE
- 15-HpETE
- Arachidonic acid
- Bezafibrate
- Daidzein
- Elafibranor
- Fonadelpar
- Genistein
- GW-0742
- GW-501516
- L-165,041
- Lanifibranor
- LG-101506
- Seladelpar
- Sodelglitazar
- Tetradecylthioacetic acid
- Antagonists: FH-535
- GSK-0660
- GSK-3787
- Agonists: 5-Oxo-ETE
- 5-Oxo-15-hydroxy-ETE
- 15-Deoxy-Δ12,14-prostaglandin J2
- 15-HETE
- 15-HpETE
- Aleglitazar
- Arachidonic acid
- Balaglitazone
- Berberine
- Bezafibrate
- Cannabidiol
- Cevoglitazar
- Chiglitazar
- Ciglitazone
- Daidzein
- Darglitazone
- Edaglitazone
- Efatutazone
- Englitazone
- Etalocib
- Farglitazar
- Genistein
- GW-1929
- Ibuprofen
- Imiglitazar
- Indeglitazar
- Lanifibranor
- LG-100268
- LG-100754
- LG-101506
- Lobeglitazone
- Muraglitazar (muroglitazar)
- nTZDpa
- Naveglitazar
- Netoglitazone
- Oxeglitazar
- Peliglitazar
- Pemaglitazar
- Perfluorononanoic acid
- Pioglitazone
- Prostaglandin J2
- Ragaglitazar
- Reglitazar
- Rivoglitazone
- Rosiglitazone
- RS5444
- Saroglitazar
- Sipoglitazar
- Sodelglitazar
- Telmisartan
- Tesaglitazar
- Troglitazone
- Antagonists: FH-535
- GW-9662
- SR-202
- T-0070907
- Unknown: SR-1664
- See also
- Receptor/signaling modulators
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